SCHEMBL28964602

SCHEMBL28964602

CC(C)(C)OC(=O)C(C)(C)COCCCCCO

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.46
CYP4F2 P78329 5/20 0.45
CYP4A11 Q02928 5/20 0.45
GAA P10253 1/20 0.39
DGAT1 O75907 1/20 0.34
ACHE P22303 6/20 0.33
MEN1 O00255 1/20 0.33
THRB P10828 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15026699 0.93 TDP1 (0.41) TDP1CYP4F2CYP4A11GAADGAT1
SCHEMBL21614510 0.85 DGAT1 (0.39) TDP1CYP4F2CYP4A11DGAT1MEN1
SCHEMBL20730298 0.84 CYP4F2 (0.46) TDP1CYP4F2CYP4A11GAAACHE
SCHEMBL16163723 0.81 MEN1 (0.42) TDP1CYP4F2CYP4A11DGAT1MEN1
SCHEMBL23971392 0.80 DGAT1 (0.31) CYP4F2CYP4A11DGAT1L3MBTL1
SCHEMBL17746739 0.77 CYP4F2 (0.61) TDP1CYP4F2CYP4A11GAADGAT1
SCHEMBL22098411 0.76 CYP4F2 (0.58) TDP1CYP4F2CYP4A11GAADGAT1
SCHEMBL23309276 0.76 CYP4F2 (0.58) TDP1CYP4F2CYP4A11GAADGAT1
SCHEMBL23673782 0.76 TDP1 (0.47) TDP1CYP4F2CYP4A11GAAACHE
SCHEMBL17941018 0.76 TDP1 (0.47) TDP1CYP4F2CYP4A11GAAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-B Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2024-04-12 CN disclosed
CN-115551862-A Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2022-12-30 CN disclosed