SCHEMBL28967191

SCHEMBL28967191

O=C(O)N1Cc2cn(-c3ccc(Br)cc3)nc2C1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.41
SLC6A9 P48067 3/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.40
PTGS2 P35354 1/20 0.38
AURKA O14965 2/20 0.36
CA12 O43570 3/20 0.36
CA9 Q16790 3/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
AKR1C3 P42330 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17202442 0.86 PDK2 (0.46) PDK2SLC6A9MEN1KMT2ANPC1
SCHEMBL29240214 0.81 MAPT (0.43) PDK2SLC6A9MEN1KMT2AHTT
SCHEMBL23015352 0.81 HDAC1 (0.45) PDK2SLC6A9
SCHEMBL29190906 0.77 HPGD (0.45) PDK2MEN1KMT2AHTTNPC1
SCHEMBL29262509 0.77 SLC6A9 (0.41) PDK2SLC6A9
SCHEMBL14861471 0.74 PDK2 (0.52) PDK2SLC6A9ALDH1A1
SCHEMBL28901850 0.74 PDK2 (0.38) PDK2SLC6A9
SCHEMBL28901868 0.74 HRH3 (0.41) PDK2SLC6A9MEN1KMT2ANPC1
SCHEMBL28967182 0.72 HPGD (0.41) PDK2SLC6A9NPC1RAB9AALDH1A1
SCHEMBL17202416 0.71 PDK2 (0.52) PDK2SLC6A9MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114667145-A Molecules that bind to TDP-43 for the treatment of amyotrophic lateral sclerosis and related disorders 拜尔哈文制药股份有限公司 2022-06-24 CN disclosed