SCHEMBL28969745

SCHEMBL28969745

O=C(O)C1=C(CF)NC2=C(C(=O)OC2)C1c1cc(F)ccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
MAPT P10636 3/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
ABCC9 O60706 11/20 0.38
KCNJ11 Q14654 11/20 0.38
ABCC8 Q09428 8/20 0.38
KCNJ8 Q15842 8/20 0.38
BRD4 O60885 1/20 0.34
BRDT Q58F21 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28969739 1.00 ALDH1A1 (0.41) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL24117102 0.89 MAPT (0.39) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969770 0.88 ALDH1A1 (0.41) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969774 0.88 ALDH1A1 (0.41) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969800 0.85 ALDH1A1 (0.41) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969763 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969760 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969787 0.82 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969769 0.81 ALDH1A1 (0.42) ALDH1A1KDM4EMAPTLMNAGAA
SCHEMBL28969773 0.81 ALDH1A1 (0.42) ALDH1A1KDM4EMAPTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115836076-A Methyl 2- (fluoromethyl) -5-oxo-4-phenyl-4,5,6,7-tetrahydro-1H-cyclopenta [ B ] pyridine-3-carboxylate and methyl 2- (fluoromethyl) -5-oxo-4-phenyl-1,4,5,7-tetrahydrofuro [3,4-B ] pyridine-3-carboxylate as CAV1.2 activators 诺华股份有限公司 2023-03-21 CN claimed
CN-115836076-A Methyl 2- (fluoromethyl) -5-oxo-4-phenyl-4,5,6,7-tetrahydro-1H-cyclopenta [ B ] pyridine-3-carboxylate and methyl 2- (fluoromethyl) -5-oxo-4-phenyl-1,4,5,7-tetrahydrofuro [3,4-B ] pyridine-3-carboxylate as CAV1.2 activators 诺华股份有限公司 2023-03-21 CN disclosed