SCHEMBL2897457

SCHEMBL2897457

CCOC(=O)CC(=O)Nc1sc(C)c(-c2ccccc2)c1C(=O)OCC

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 15/20 0.69
LMNA P02545 7/20 0.69
THRB P10828 5/20 0.69
HTT P42858 4/20 0.69
GAA P10253 1/20 0.66
MAPT P10636 9/20 0.64
MEN1 O00255 4/20 0.64
KMT2A Q03164 4/20 0.64
HPGD P15428 5/20 0.61
SMN1; SMN2 Q16637 5/20 0.61
KDM4E B2RXH2 2/20 0.61
PTBP1 P26599 1/20 0.61
TDP1 Q9NUW8 1/20 0.60
NPSR1 Q6W5P4 5/20 0.56
POLB P06746 1/20 0.54
MAPK1 P28482 1/20 0.54
RECQL P46063 1/20 0.54
ATM Q13315 1/20 0.54
CYP3A4 P08684 2/20 0.53
CYP2C19 P33261 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3611687 0.92 ALDH1A1 (0.57) ALDH1A1LMNATHRBHTTGAA
SCHEMBL13837687 0.86 ALDH1A1 (0.73) ALDH1A1LMNATHRBHTTGAA
SCHEMBL3472339 0.81 ALDH1A1 (1.00) ALDH1A1LMNATHRBHTTGAA
SCHEMBL3472335 0.81 ALDH1A1 (1.00) ALDH1A1LMNATHRBHTTGAA
SCHEMBL12851713 0.81 ALDH1A1 (0.85) ALDH1A1LMNATHRBHTTGAA
SCHEMBL8051335 0.80 ALDH1A1 (0.64) ALDH1A1LMNATHRBHTTGAA
SCHEMBL8051341 0.80 ALDH1A1 (0.64) ALDH1A1LMNATHRBHTTGAA
SCHEMBL2897094 0.79 POLB (0.74) ALDH1A1LMNAHTTGAAMAPT
SCHEMBL3913084 0.77 ALDH1A1 (0.55) ALDH1A1LMNATHRBHTTGAA
SCHEMBL3935830 0.77 ALDH1A1 (0.60) ALDH1A1LMNATHRBHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879899-B1 THIENOPYRIDINE DERIVATIVES AS POTASSIUM CHANNEL INHIBITORS XENTION LTD (GB) 2010-08-04 EP disclosed