SCHEMBL28974972

SCHEMBL28974972

Cc1cc(-c2c(C(C)C)c(NC(C)C(=O)O)nc3cc(O)ccc23)ccc1F

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 10/20 0.37
MCL1 Q07820 3/20 0.35
BCL2 P10415 2/20 0.35
BCL2L1 Q07817 1/20 0.35
KCNQ3 O43525 3/20 0.34
KCNQ2 O43526 3/20 0.34
CYP2C9 P11712 3/20 0.34
TOP1 P11387 1/20 0.33
APP P05067 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23895822 1.00 PDE10A (0.37) PDE10AMCL1BCL2BCL2L1KCNQ3
SCHEMBL25544154 1.00 PDE10A (0.37) PDE10AMCL1BCL2BCL2L1KCNQ3
SCHEMBL25558990 0.91 PDE10A (0.38) PDE10AMCL1BCL2BCL2L1KCNQ3
SCHEMBL23896035 0.91 PDE10A (0.38) PDE10AMCL1BCL2BCL2L1KCNQ3
SCHEMBL23896036 0.91 PDE10A (0.38) PDE10AMCL1BCL2BCL2L1KCNQ3
SCHEMBL23895820 0.89 TRPV3 (0.35) PDE10AMCL1BCL2L1KCNQ3KCNQ2
SCHEMBL25544155 0.89 TRPV3 (0.35) PDE10AMCL1BCL2L1KCNQ3KCNQ2
SCHEMBL23896419 0.89 CTSA (0.35) KCNQ3KCNQ2TOP1
SCHEMBL23896415 0.89 CTSA (0.35) KCNQ3KCNQ2TOP1
SCHEMBL23896209 0.88 SCN9A (0.39) PDE10AMCL1BCL2BCL2L1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115697969-A 7-or 8-hydroxy-isoquinoline and 7-or 8-hydroxy-quinoline derivatives as alpha-1 antitrypsin modulators for the treatment of alpha-1 antitrypsin deficiency (AATD) 弗特克斯药品有限公司 2023-02-03 CN disclosed