SCHEMBL28977161

SCHEMBL28977161

CN1CCN(c2ccc(-c3cc(-c4ccc(OCc5ccccc5)c(C(F)(F)F)c4)n[nH]3)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.60
PRKD1 Q15139 9/20 0.52
HTR6 P50406 2/20 0.48
MAP4K1 Q92918 2/20 0.48
FLT1 P17948 2/20 0.46
KDR P35968 2/20 0.46
FLT3 P36888 2/20 0.46
AURKA O14965 1/20 0.45
CTSS P25774 2/20 0.44
ALK Q9UM73 2/20 0.43
CTSK P43235 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28977180 0.88 MELK (0.64) MELKPRKD1HTR6MAP4K1FLT1
SCHEMBL28977160 0.88 MELK (0.57) MELKPRKD1MAP4K1CTSSCTSK
SCHEMBL28977164 0.87 MELK (0.65) MELKPRKD1HTR6MAP4K1FLT1
SCHEMBL28977194 0.85 MAP4K1 (0.61) MELKPRKD1MAP4K1
SCHEMBL28977181 0.83 MELK (0.73) MELKPRKD1MAP4K1FLT1KDR
SCHEMBL28977166 0.81 MELK (0.65) MELKPRKD1HTR6MAP4K1FLT1
SCHEMBL28687893 0.80 MAP4K1 (0.57) HTR6MAP4K1ALK
SCHEMBL30290614 0.80 MAP4K1 (0.57) HTR6MAP4K1ALK
SCHEMBL28977172 0.75 MELK (0.86) MELKPRKD1MAP4K1KDRFLT3
SCHEMBL28977189 0.75 MELK (0.73) MELKPRKD1MAP4K1KDRFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113861188-B Pyrazolo [3,4-b ] pyridine derivative, preparation method thereof and application thereof as HPK1 inhibitor 杭州医学院 2023-02-28 CN disclosed