SCHEMBL28977181

SCHEMBL28977181

CN1CCN(c2ccc(-c3cc(-c4ccc(OCc5ccccc5)cc4)n[nH]3)cc2)CC1

nearest known ligand 0.73

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.73
MAP4K1 Q92918 1/20 0.62
PRMT5 O14744 3/20 0.56
ALK Q9UM73 1/20 0.54
PRKD1 Q15139 9/20 0.52
FLT3 P36888 4/20 0.51
FLT1 P17948 2/20 0.51
KDR P35968 2/20 0.51
KIT P10721 1/20 0.51
AURKA O14965 1/20 0.50
NPC1 O15118 1/20 0.50
TP53 P04637 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28977166 0.86 MELK (0.65) MELKMAP4K1PRMT5ALKPRKD1
SCHEMBL28977164 0.86 MELK (0.65) MELKMAP4K1PRMT5ALKPRKD1
SCHEMBL28977167 0.86 MELK (0.70) MELKMAP4K1PRKD1FLT3KDR
SCHEMBL28977180 0.85 MELK (0.64) MELKMAP4K1PRMT5ALKPRKD1
SCHEMBL28977192 0.83 MELK (0.66) MELKMAP4K1PRKD1NPC1TP53
SCHEMBL28977161 0.83 MELK (0.60) MELKMAP4K1ALKPRKD1FLT3
SCHEMBL13202898 0.82 RAB9A (0.67) MAP4K1PRMT5ALKNPC1TP53
SCHEMBL28977159 0.79 MELK (0.82) MELKMAP4K1PRKD1FLT3KDR
SCHEMBL28977165 0.79 MELK (0.70) MELKMAP4K1PRKD1FLT3FLT1
SCHEMBL28977172 0.79 MELK (0.86) MELKMAP4K1ALKPRKD1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113861188-B Pyrazolo [3,4-b ] pyridine derivative, preparation method thereof and application thereof as HPK1 inhibitor 杭州医学院 2023-02-28 CN disclosed