SCHEMBL28977403

SCHEMBL28977403

C#Cc1ccc(C(C)n2cnc3c(N)ncnc32)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.57
ADORA1 P30542 3/20 0.57
ADORA2B P29275 2/20 0.57
PI4KA P42356 1/20 0.57
PI4K2B Q8TCG2 1/20 0.57
PI4K2A Q9BTU6 1/20 0.57
PI4KB Q9UBF8 1/20 0.57
ADA P00813 4/20 0.43
PIK3CD O00329 2/20 0.43
PDE2A O00408 2/20 0.43
CYP3A4 P08684 2/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX15 P16050 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23977342 1.00 ADORA2A (0.57) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL30291134 1.00 ADORA2A (0.57) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL13269011 0.82 ADORA2A (0.65) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL13268766 0.82 ADORA2A (0.65) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL28977406 0.78 HTR2C (0.46) PIK3CD
SCHEMBL30225391 0.78 HTR2C (0.46) PIK3CD
SCHEMBL23977241 0.78 HTR2C (0.46) PIK3CD
SCHEMBL30225397 0.75 TDP1 (0.38) PIK3CD
SCHEMBL754007 0.74 ADORA2A (1.00) ADORA2AADORA1ADORA2BPI4KAPI4K2B
Hydrochloric Acid SCHEMBL30881556 0.73 ADORA2A (0.96) ADORA2AADORA1ADORA2BPI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4143172-A1 ANTIBACTERIAL AND ANTIFUNGAL PLEUROMUTILIN CONJUGATES Syddansk Universitet (DK) 2023-03-08 EP disclosed
CN-115720579-A Antibacterial and antifungal pleuromutilin conjugates 赛丹思科大学 2023-02-28 CN disclosed