SCHEMBL289794

SCHEMBL289794

Clc1csc(-c2cccnc2)n1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.67
AXL P30530 1/20 0.67
PBRM1 Q86U86 1/20 0.67
MKNK1 Q9BUB5 1/20 0.67
MKNK2 Q9HBH9 1/20 0.67
CYP2E1 P05181 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2A6 P11509 1/20 0.65
CYP2C9 P11712 1/20 0.65
CYP2B6 P20813 1/20 0.65
RAB9A P51151 4/20 0.63
KDM4E B2RXH2 3/20 0.63
ALDH1A1 P00352 2/20 0.63
HPGD P15428 2/20 0.60
CASP3 P42574 1/20 0.60
SENP8 Q96LD8 1/20 0.60
SENP7 Q9BQF6 1/20 0.60
SENP6 Q9GZR1 1/20 0.60
NPC1 O15118 2/20 0.58
HSD17B10 Q99714 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6196239 0.80 CYP19A1 (1.00) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL28232733 0.79 KDM4E (0.59) CYP19A1RAB9AKDM4EHPGDNPC1
SCHEMBL27820489 0.79 KDM4E (0.53) CYP19A1RAB9AKDM4EALDH1A1HPGD
SCHEMBL266591 0.79 CYP2E1 (1.00) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL9829144 0.79 CYP19A1 (0.67) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL14359963 0.79 CYP19A1 (0.67) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL1722906 0.79 CYP19A1 (0.67) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL12402375 0.79 CYP19A1 (0.67) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL5377137 0.78 CYP19A1 (0.61) CYP19A1AXLPBRM1MKNK1MKNK2
SCHEMBL21408714 0.78 CYP19A1 (0.40) CYP19A1AXLPBRM1MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9756858-B2 Insecticides SYNGENTA PARTICIPATIONS AG (CH) 2017-09-12 US disclosed
US-9756858-B2 Insecticides SYNGENTA PARTICIPATIONS AG (CH) 2017-09-12 US disclosed
US-9756858-B2 Insecticides SYNGENTA PARTICIPATIONS AG (CH) 2017-09-12 US disclosed
CN-104540821-B Process for preparing certain 2- (pyridin-3-yl) thiazoles 美国陶氏益农公司 2017-07-18 CN disclosed
EP-2614826-B1 Process for preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2017-03-01 EP disclosed
EP-2614826-B1 Process for preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2017-03-01 EP disclosed
US-9357780-B2 Pesticidal compositions DOW AGROSCIENCES LLC (US) 2016-06-07 US disclosed
US-9357780-B2 Pesticidal compositions DOW AGROSCIENCES LLC (US) 2016-06-07 US disclosed
US-9357780-B2 Pesticidal compositions DOW AGROSCIENCES LLC (US) 2016-06-07 US disclosed
EP-2614825-B1 Process for the preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2016-03-16 EP disclosed
WO-2012168361-A1 NOVEL INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-12-13 WO disclosed
EP-2532661-A1 Novel insecticides Syngenta Participations AG (CH) 2012-12-12 EP disclosed
EP-2532661-A1 Novel insecticides Syngenta Participations AG (CH) 2012-12-12 EP disclosed
CN-102458403-A insecticidal composition DOW AGROSCIENCES LLC 2012-05-16 CN disclosed
EP-2427191-A1 PESTICIDAL COMPOSITIONS Dow AgroSciences LLC (US) 2012-03-14 EP disclosed
US-20100292253-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-18 US disclosed
US-20100292253-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-18 US disclosed
US-20100292253-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-18 US disclosed
WO-2010129497-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-11 WO disclosed
WO-2010129497-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100292253-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 CYP19A1 234/4885AXL 4147/4885PBRM1 4590/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.