SCHEMBL28979421

SCHEMBL28979421

COc1cc2ncnc(Oc3ccc(C(=O)C(N)=O)cc3)c2cc1OC

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.65
PDGFRA P16234 1/20 0.64
CSF1R P07333 1/20 0.61
MET P08581 2/20 0.61
AURKA O14965 1/20 0.61
TEK Q02763 1/20 0.61
AURKB Q96GD4 1/20 0.61
PDGFRB P09619 3/20 0.58
FLT4 P35916 3/20 0.58
RET P07949 1/20 0.57
KIF5B P33176 1/20 0.57
LCK P06239 1/20 0.56
PDE10A Q9Y233 1/20 0.56
RAF1 P04049 1/20 0.55
KIT P10721 1/20 0.55
SRC P12931 1/20 0.55
FLT1 P17948 1/20 0.55
EGFR P00533 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30448125 1.00 KDR (0.65) KDRPDGFRACSF1RMETAURKA
SCHEMBL14967551 0.90 KDR (0.67) KDRPDGFRACSF1RMETAURKA
SCHEMBL30447769 0.89 KDR (0.66) KDRPDGFRACSF1RMETAURKA
SCHEMBL28468402 0.89 KDR (0.66) KDRPDGFRACSF1RMETAURKA
SCHEMBL28464530 0.84 KDR (0.69) KDRPDGFRACSF1RPDGFRBFLT4
SCHEMBL30448369 0.84 KDR (0.69) KDRPDGFRACSF1RPDGFRBFLT4
SCHEMBL30448257 0.82 KDR (0.78) KDRPDGFRACSF1RMETPDGFRB
SCHEMBL5177524 0.82 PDGFRB (0.66) KDRPDGFRACSF1RMETAURKA
SCHEMBL28470525 0.82 KDR (0.66) KDRPDGFRACSF1RMETAURKA
SCHEMBL28474029 0.81 KDR (0.58) KDRPDGFRACSF1RMETAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825605-B Aryl ketone amide compound and preparation method and application thereof 中国科学院上海药物研究所 2023-03-31 CN disclosed