SCHEMBL28979780

SCHEMBL28979780

O=C1NC(=O)C(F)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.48
CASP3 P42574 2/20 0.42
CASP7 P55210 2/20 0.42
CASP6 P55212 2/20 0.42
CASP8 Q14790 2/20 0.42
CASP2 P42575 1/20 0.42
PDGFRA P16234 1/20 0.41
FER P16591 1/20 0.41
LTK P29376 1/20 0.41
CDK8 P49336 1/20 0.41
ACVR1 Q04771 1/20 0.41
LRRK2 Q5S007 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
PARP1 P09874 3/20 0.39
TNKS2 Q9H2K2 3/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
HSD17B10 Q99714 3/20 0.38
TDP2 O95551 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30521243 0.81 TNKS2 (0.37) GSK3BCASP3CASP7CASP6CASP8
SCHEMBL11844924 0.78 GSK3B (0.50) GSK3BCASP3CASP7CASP6CASP8
SCHEMBL2337529 0.76 GSK3B (0.48) GSK3BCASP3CASP7CASP6CASP8
SCHEMBL5551044 0.76 GSK3B (0.48) GSK3BCASP3CASP7CASP6CASP8
SCHEMBL31362875 0.76 GSK3B (0.43) GSK3BCASP3CASP7CASP6CASP8
SCHEMBL30364585 0.75 IDO1 (0.50) GSK3BPARP1L3MBTL1KDM4EALDH1A1
SCHEMBL5144419 0.75 IDO1 (0.50) GSK3BPARP1L3MBTL1KDM4EALDH1A1
SCHEMBL17434393 0.72 GSK3B (0.43) GSK3BCASP3CASP7CASP6CASP8
SCHEMBL19926520 0.72 MEN1 (0.42) TNKS2HTR2BTDP2MAOAMAOB
SCHEMBL11801695 0.71 HSD17B10 (0.47) GSK3BCASP3CASP7CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115747843-B Electrochemical preparation method for synthesizing fluoroisoquinoline-1, 3-diketone compound by trifluoromethyl/cyclization 兰州石化职业技术大学 2025-01-24 CN claimed
CN-115747843-A Electrochemical preparation method for synthesizing fluoroisoquinoline-1,3-diketone compound through trifluoromethylation/cyclization 兰州石化职业技术大学 2023-03-07 CN claimed
CN-115747843-B Electrochemical preparation method for synthesizing fluoroisoquinoline-1, 3-diketone compound by trifluoromethyl/cyclization 兰州石化职业技术大学 2025-01-24 CN disclosed
WO-2023143494-A1 NEW PROTAC COMPOUND 甘李药业股份有限公司 2023-08-03 WO disclosed