SCHEMBL28980964

SCHEMBL28980964

CC(=O)Nc1ccc(Nc2nc(Nc3ccc(N4CCN(C)CC4)cc3)ncc2Cl)cc1Cl

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K7 O43318 4/20 0.72
ALK Q9UM73 4/20 0.69
WEE1 P30291 2/20 0.69
CDK9 P50750 2/20 0.66
CCNT1 O60563 1/20 0.66
CCNK O75909 1/20 0.66
CYP3A4 P08684 1/20 0.66
CCND3 P30281 1/20 0.66
CDK6 Q00534 1/20 0.66
BRD4 O60885 9/20 0.66
FGFR1 P11362 2/20 0.65
MAP2K1 Q02750 2/20 0.65
SRC P12931 1/20 0.65
MAPK1 P28482 1/20 0.65
SLC2A1 P11166 1/20 0.64
CHEK1 O14757 1/20 0.64
AURKA O14965 1/20 0.64
DAPK3 O43293 1/20 0.64
JAK2 O60674 1/20 0.64
PRKD3 O94806 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31684799 1.00 MAP3K7 (0.72) MAP3K7ALKWEE1CDK9CCNT1
SCHEMBL28981000 0.93 BRD4 (0.66) MAP3K7ALKWEE1CDK9CCNT1
SCHEMBL31684797 0.93 BRD4 (0.66) MAP3K7ALKWEE1CDK9CCNT1
SCHEMBL28980963 0.90 ALK (0.68) MAP3K7ALKWEE1CDK9CCNT1
SCHEMBL31684751 0.90 ALK (0.68) MAP3K7ALKWEE1CDK9CCNT1
SCHEMBL28980993 0.90 MAP3K7 (0.65) MAP3K7ALKWEE1CDK9BRD4
SCHEMBL28980991 0.90 MAP3K7 (0.70) MAP3K7ALKWEE1CDK9BRD4
SCHEMBL31684761 0.90 MAP3K7 (0.65) MAP3K7ALKWEE1CDK9BRD4
SCHEMBL31684780 0.90 MAP3K7 (0.70) MAP3K7ALKWEE1CDK9BRD4
SCHEMBL31684777 0.90 MAP3K7 (0.80) MAP3K7ALKBRD4FGFR1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN claimed
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN disclosed