SCHEMBL28980986

SCHEMBL28980986

C=CC(=O)Nc1ccc(Nc2nc(Nc3ccc(N4CCN(C)CC4)cn3)ncc2Cl)cc1Cl

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCND3 P30281 12/20 0.69
CDK6 Q00534 12/20 0.69
CCNK O75909 11/20 0.69
CDK9 P50750 11/20 0.69
CYP3A4 P08684 2/20 0.69
CCNT1 O60563 1/20 0.69
MAP3K7 O43318 5/20 0.68
MAP2K1 Q02750 4/20 0.68
MAPK1 P28482 2/20 0.68
FGFR1 P11362 1/20 0.68
SRC P12931 1/20 0.68
CCNA2 P20248 2/20 0.63
CDK2 P24941 2/20 0.63
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
CTSC P53634 1/20 0.61
FLT3 P36888 1/20 0.59
JAK3 P52333 1/20 0.57
BTK Q06187 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31684756 1.00 CCND3 (0.69) CCND3CDK6CCNKCDK9CYP3A4
SCHEMBL31684777 0.91 MAP3K7 (0.80) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL28980982 0.91 MAP3K7 (0.80) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL28980998 0.88 MAP3K7 (0.73) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL31684766 0.88 MAP3K7 (0.73) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL31684785 0.85 MAP3K7 (0.66) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL28980978 0.85 MAP3K7 (0.66) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL31684776 0.85 MAP3K7 (0.70) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL28980973 0.85 MAP3K7 (0.70) MAP3K7MAP2K1MAPK1FGFR1SRC
SCHEMBL31684746 0.84 JAK3 (0.71) MAP3K7MAP2K1MAPK1FGFR1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN claimed
CN-115894381-A 2,4,5-trisubstituted pyrimidine compound and preparation method and application thereof 温州医科大学 2023-04-04 CN disclosed