SCHEMBL28984043

SCHEMBL28984043

CCOC(=O)c1cc(Br)n(C)c1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.47
KMT2A Q03164 3/20 0.47
GAA P10253 2/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPK1 P28482 1/20 0.46
BAZ2B Q9UIF8 1/20 0.45
BAZ2A Q9UIF9 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11359782 0.82 TSHR (0.56) TSHRKMT2AGAAMAPTPKM
SCHEMBL23732187 0.79 TSHR (0.47) TSHRKMT2AGAAMAPTALDH1A1
SCHEMBL14830469 0.79 KDM4E (0.47) TSHRKMT2AGAAMAPTALDH1A1
SCHEMBL15568745 0.78 KMT2A (0.34) KMT2AGAAMAPTPKMALDH1A1
SCHEMBL1220842 0.78 ALDH1A1 (0.52) TSHRKMT2AGAAMAPTALDH1A1
SCHEMBL27077665 0.78 TSHR (0.49) TSHRKMT2AGAAMAPTALDH1A1
SCHEMBL26088044 0.77 KMT2A (0.48) TSHRKMT2AGAAMAPTALDH1A1
SCHEMBL12854715 0.77 TSHR (0.48) TSHRKMT2AGAAALDH1A1KDM4E
SCHEMBL21408332 0.76 NPSR1 (0.45) TSHRKMT2AGAAMAPTALDH1A1
SCHEMBL21408425 0.76 NPSR1 (0.48) TSHRKMT2AGAAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115960083-A Heterocyclic compounds, their preparation and use 百极弘烨(南通)医药科技有限公司 2023-04-14 CN disclosed