SCHEMBL28989403

SCHEMBL28989403

COc1cc(Br)ccc1CC(NC(=O)OC(C)(C)C)C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 9/20 0.47
CTSS P25774 4/20 0.45
CTSK P43235 4/20 0.45
CTSB P07858 1/20 0.44
REN P00797 2/20 0.43
TACR1 P25103 1/20 0.43
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
CACNA1B Q00975 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26781565 1.00 AAK1 (0.47) AAK1CTSSCTSKCTSBREN
SCHEMBL28989419 0.90 TACR1 (0.48) AAK1CTSSCTSKCTSBTACR1
SCHEMBL24981981 0.90 TACR1 (0.48) AAK1CTSSCTSKCTSBTACR1
SCHEMBL24981983 0.90 ACE (0.49) AAK1CTSSCTSKCTSBTACR1
SCHEMBL28989259 0.90 ACE (0.49) AAK1CTSSCTSKCTSBTACR1
SCHEMBL19858738 0.85 AAK1 (0.51) AAK1CTSSCTSKCTSBREN
SCHEMBL30476240 0.85 AAK1 (0.51) AAK1CTSSCTSKCTSBREN
SCHEMBL16035979 0.85 AAK1 (0.51) AAK1CTSSCTSKCTSBREN
SCHEMBL20661656 0.83 TACR1 (0.59) CTSSCTSKCTSBRENTACR1
SCHEMBL14974873 0.83 TACR1 (0.59) CTSSCTSKCTSBRENTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996923-A Nitrile derivative as dipeptidyl peptidase 1 inhibitor and application thereof 四川海思科制药有限公司 2023-04-21 CN disclosed