SCHEMBL28989259

SCHEMBL28989259

COc1cc(Br)ccc1CC(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.49
CTSS P25774 4/20 0.48
CTSK P43235 4/20 0.48
ITGA4 P13612 2/20 0.48
ITGB7 P26010 2/20 0.48
CTSB P07858 1/20 0.47
SCN9A Q15858 1/20 0.47
AAK1 Q2M2I8 5/20 0.46
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
TACR1 P25103 1/20 0.44
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
PTPN1 P18031 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24981983 1.00 ACE (0.49) ACECTSSCTSKITGA4ITGB7
SCHEMBL24981981 0.91 TACR1 (0.48) CTSSCTSKCTSBAAK1TACR1
SCHEMBL28989419 0.91 TACR1 (0.48) CTSSCTSKCTSBAAK1TACR1
SCHEMBL3553358 0.91 ACE (0.49) ACECTSSCTSKITGA4ITGB7
SCHEMBL21243764 0.91 ACE (0.49) ACECTSSCTSKITGA4ITGB7
SCHEMBL30829404 0.91 ACE (0.49) ACECTSSCTSKITGA4ITGB7
SCHEMBL3553357 0.91 ACE (0.49) ACECTSSCTSKITGA4ITGB7
SCHEMBL28989403 0.90 AAK1 (0.47) CTSSCTSKCTSBAAK1TACR1
SCHEMBL26781565 0.90 AAK1 (0.47) CTSSCTSKCTSBAAK1TACR1
SCHEMBL8650368 0.87 SCN9A (0.52) ACECTSSCTSKITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996923-A Nitrile derivative as dipeptidyl peptidase 1 inhibitor and application thereof 四川海思科制药有限公司 2023-04-21 CN disclosed