SCHEMBL28996233

SCHEMBL28996233

Cc1ncc(Cl)nc1-c1nc(-c2nccs2)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.43
RAB9A P51151 1/20 0.39
SYK P43405 5/20 0.36
SRC P12931 4/20 0.36
ZAP70 P43403 3/20 0.36
ADORA2A P29274 3/20 0.35
ADORA1 P30542 2/20 0.35
CYP1A1 P04798 3/20 0.34
CYP1A2 P05177 3/20 0.34
CYP1B1 Q16678 3/20 0.34
CDK2 P24941 1/20 0.34
HPGD P15428 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
PKMYT1 Q99640 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
PDE10A Q9Y233 2/20 0.33
SPHK2 Q9NRA0 1/20 0.33
SPHK1 Q9NYA1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30252995 0.82 ADORA2A (0.39) HSP90AA1SYKSRCZAP70ADORA2A
SCHEMBL28996009 0.82 ADORA2A (0.39) HSP90AA1SYKSRCZAP70ADORA2A
SCHEMBL30253005 0.79 HSP90AA1 (0.38) HSP90AA1SYKSRCZAP70ADORA2A
SCHEMBL28996098 0.79 HSP90AA1 (0.38) HSP90AA1SYKSRCZAP70ADORA2A
SCHEMBL2185378 0.73 HSP90AA1 (0.57) HSP90AA1RAB9ASYKSRCZAP70
SCHEMBL28996033 0.68 ADORA2A (0.39) HSP90AA1SYKSRCZAP70ADORA2A
SCHEMBL30252594 0.68 ADORA2A (0.39) HSP90AA1SYKSRCZAP70ADORA2A
SCHEMBL319118 0.63 HSP90AA1 (0.51) HSP90AA1RAB9ASYKADORA2AADORA1
SCHEMBL29290792 0.63 RAB9A (0.51) HSP90AA1RAB9ASYKSRCZAP70
SCHEMBL320331 0.62 HSP90AA1 (0.47) HSP90AA1RAB9ASYKSRCZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed