SCHEMBL289986

SCHEMBL289986

N#CC(Cc1ccc(-c2ccc(F)cc2)cc1)C1CC(C(N)=O)CCO1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSC P53634 7/20 0.42
DPP4 P27487 8/20 0.41
DPP8 Q6V1X1 4/20 0.37
DPP9 Q86TI2 4/20 0.37
DPP7 Q9UHL4 3/20 0.37
FAP Q12884 3/20 0.37
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
MAOB P27338 1/20 0.34
ACACB O00763 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290171 0.90 CTSC (0.45) CTSC
SCHEMBL289949 0.89 CTSC (0.44) CTSC
SCHEMBL290044 0.89 CTSC (0.44) CTSCDPP4DPP8DPP9DPP7
SCHEMBL290338 0.87 CTSC (0.44) CTSCDPP4DPP8DPP9DPP7
SCHEMBL290567 0.81 CTSC (0.51) CTSC
SCHEMBL288811 0.80 CTSC (0.49) CTSCDPP4ACACB
SCHEMBL289369 0.79 CTSC (0.53) CTSC
SCHEMBL289754 0.79 CTSC (0.52) CTSC
SCHEMBL299868 0.78 CTSC (0.47) CTSC
SCHEMBL299206 0.78 CTSC (0.53) CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP claimed
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed