SCHEMBL299206

SCHEMBL299206

CN1C(=O)COc2ccc(-c3ccc(CC(C#N)C4CC(C(N)=O)CCO4)cc3)cc21

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSC P53634 18/20 0.53
CTSK P43235 2/20 0.39
USP30 Q70CQ3 1/20 0.38
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289369 0.87 CTSC (0.53) CTSCCTSK
SCHEMBL299868 0.84 CTSC (0.47) CTSCCTSKPDE3BPDE3A
SCHEMBL289754 0.79 CTSC (0.52) CTSCCTSK
SCHEMBL290171 0.78 CTSC (0.45) CTSCCTSK
SCHEMBL289986 0.78 CTSC (0.42) CTSC
SCHEMBL289949 0.78 CTSC (0.44) CTSCCTSK
SCHEMBL290338 0.77 CTSC (0.44) CTSC
SCHEMBL299207 0.77 CTSC (0.69) CTSCCTSK
SCHEMBL290567 0.76 CTSC (0.51) CTSCCTSK
SCHEMBL290044 0.75 CTSC (0.44) CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP claimed
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed