SCHEMBL289992

SCHEMBL289992

Cc1c(F)c(F)cc(C#N)c1F

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 3/20 0.43
KHK P50053 1/20 0.37
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
CYP11B1 P15538 3/20 0.35
CYP11B2 P19099 3/20 0.35
EGLN2 Q96KS0 2/20 0.33
TSHR P16473 1/20 0.33
AR P10275 5/20 0.33
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16127310 0.88 TRPV4 (0.38) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL27362042 0.86 TRPV4 (0.43) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL10474330 0.83 KHK (0.43) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL3191461 0.82 TRPV4 (0.43) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL30493379 0.82 TRPV4 (0.43) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL25436881 0.82 TRPV4 (0.43) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL23010977 0.82 TSHR (0.38) TRPV4ESR1ESR2CYP11B1CYP11B2
SCHEMBL17687703 0.81 KHK (0.42) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL17687678 0.81 TRPV4 (0.39) TRPV4KHKESR1ESR2CYP11B1
SCHEMBL19780236 0.81 ESR1 (0.40) TRPV4KHKESR1ESR2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116003253-A Preparation method of trifluoro-phenylpyrimidine intermediate 2- [3- (trifluoromethyl) phenyl ] dimethyl malonate 上海试四化学品有限公司 2023-04-25 CN claimed
US-20040110990-A1 Catalytic reduction of nitriles to aldehydes LANXESS DEUTSCHLAND GMBH (DE) 2004-06-10 US claimed
EP-2427801-A1 FUNCTIONALIZED PERFLUOROPOLYETHER MATERIAL AS A HYDROPHOBIC COATING Hewlett-Packard Development Company, L.P. (US) 2012-03-14 EP disclosed
WO-2010128969-A1 FUNCTIONALIZED PERFLUOROPOLYETHER MATERIAL AS A HYDROPHOBIC COATING HEWLETT-PACKARD DEVELOPMENT COMPANY, L.P. (US) 2010-11-11 WO disclosed
US-6784308-B2 CATALYZING THE NITRIDING REACTION OF HALOGENOAROMATICS OR ARYL PERFLUOROSULFONATES AND ALKALI METAL CYANIDES BAYER AKTIENGESELLSCHAFT (DE) 2004-08-31 US disclosed
EP-0237955-B1 QUINOLONECARBOXYLIC ACID DERIVATIVES AND THEIR PREPARATION KYORIN PHARMACEUTICAL CO., LTD. (JP) 1992-07-15 EP disclosed
US-4894458-A BACTERICIDES KYORIN PHARMACEUTICAL CO., LTD. (JP) 1990-01-16 US disclosed
EP-0237955-A2 Quinolonecarboxylic acid derivatives and their preparation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1987-09-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040110990-A1 Catalytic reduction of nitriles to aldehydes CAT, NIT2, IDH1 TRPV4 2019/4885KHK 1274/4885ESR1 2389/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.