SCHEMBL29004707

SCHEMBL29004707

CC(C)c1n[nH]c2nccc(Br)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.39
PRKCI P41743 1/20 0.37
LRRK2 Q5S007 4/20 0.33
AURKA O14965 1/20 0.32
DAPK3 O43293 1/20 0.32
JAK2 O60674 1/20 0.32
MAP4K4 O95819 1/20 0.32
PAK4 O96013 1/20 0.32
ABL1 P00519 1/20 0.32
LCK P06239 1/20 0.32
FYN P06241 1/20 0.32
CSF1R P07333 1/20 0.32
RET P07949 1/20 0.32
IGF1R P08069 1/20 0.32
FLT1 P17948 1/20 0.32
LTK P29376 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30332332 1.00 DAO (0.39) DAOPRKCILRRK2AURKADAPK3
SCHEMBL27010940 0.81 LRRK2 (0.34) LRRK2AURKADAPK3JAK2MAP4K4
SCHEMBL2691540 0.79 AURKB (0.41) DAOPRKCILRRK2AURKADAPK3
SCHEMBL30332245 0.79 LRRK2 (0.33) LRRK2AURKADAPK3JAK2MAP4K4
SCHEMBL30332414 0.79 AURKB (0.41) DAOPRKCILRRK2AURKADAPK3
SCHEMBL2693015 0.79 LRRK2 (0.33) LRRK2AURKADAPK3JAK2MAP4K4
SCHEMBL26661511 0.77 LRRK2 (0.32) LRRK2AURKADAPK3JAK2MAP4K4
SCHEMBL29767999 0.77 PRKCI (0.40) DAOPRKCILRRK2
SCHEMBL29079633 0.77 PRKCI (0.40) DAOPRKCILRRK2
SCHEMBL25245801 0.76 PRKCI (0.42) DAOPRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115960100-B Synthesis method of Pi Mite xib drug for treating gastrointestinal stromal tumor 北京康立生医药技术开发有限公司 2023-08-18 CN disclosed
CN-115960100-A Synthetic method of drug Pi Mite Xibu for treating gastrointestinal stromal tumor 北京康立生医药技术开发有限公司 2023-04-14 CN disclosed