SCHEMBL29008571

SCHEMBL29008571

O=CN1Cc2cccc(N3CCCC(O)C3)c2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 1/20 0.39
SMARCA4 P51532 1/20 0.39
PBRM1 Q86U86 1/20 0.39
CHRM2 P08172 2/20 0.38
CHRM4 P08173 2/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 1/20 0.38
TIPARP Q7Z3E1 1/20 0.38
DRD3 P35462 3/20 0.38
HTR6 P50406 3/20 0.38
DRD2 P14416 1/20 0.38
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CCNE2 O96020 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
TSHR P16473 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24913825 0.74 SMARCA2 (0.39) SMARCA2SMARCA4PBRM1CHRM2CHRM4
SCHEMBL31062432 0.74 SMARCA2 (0.39) SMARCA2SMARCA4PBRM1CHRM2CHRM4
Hydrochloric Acid SCHEMBL30368686 0.73 SMARCA2 (0.39) SMARCA2SMARCA4PBRM1CHRM2CHRM4
Hydrochloric Acid SCHEMBL29008605 0.73 SMARCA2 (0.39) SMARCA2SMARCA4PBRM1CHRM2CHRM4
SCHEMBL9367057 0.70 NOTUM (0.55) SMARCA2SMARCA4PBRM1LMNAALDH1A1
SCHEMBL15896058 0.70 KDM4E (0.46) SMARCA2SMARCA4PBRM1ALDH1A1CCNE2
SCHEMBL29823001 0.70 KDM4E (0.46) SMARCA2SMARCA4PBRM1ALDH1A1CCNE2
SCHEMBL3435118 0.69 KEAP1 (0.58) SMARCA2SMARCA4PBRM1CHRM2CHRM4
SCHEMBL30783767 0.69 SMARCA2 (0.47) SMARCA2SMARCA4PBRM1CHRM2CHRM4
SCHEMBL30784053 0.69 SMARCA2 (0.47) SMARCA2SMARCA4PBRM1CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117693507-A Inhibitor compounds 奈奥芬莱有限公司 2024-03-12 CN claimed
CN-115996907-A Inhibitors of MLH1 and/or PMS2 for cancer treatment 奈奥芬莱有限公司 2023-04-21 CN claimed
CN-117693507-A Inhibitor compounds 奈奥芬莱有限公司 2024-03-12 CN disclosed
CN-115996907-A Inhibitors of MLH1 and/or PMS2 for cancer treatment 奈奥芬莱有限公司 2023-04-21 CN disclosed