SCHEMBL29010959

SCHEMBL29010959

Nc1ccc2c(c1)C(=O)N(Cc1ccccc1)C2

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 1/20 0.55
HPGD P15428 1/20 0.55
HDAC1 Q13547 5/20 0.55
HDAC4 P56524 3/20 0.55
HDAC6 Q9UBN7 3/20 0.55
PARP1 P09874 1/20 0.48
DHPS P49366 1/20 0.45
ACHE P22303 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
GRM5 P41594 1/20 0.43
NR3C1 P04150 1/20 0.43
PREP P48147 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
CRBN Q96SW2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31391661 1.00 KDM4E (0.55) KDM4EALDH1A1HPGDHDAC1HDAC4
SCHEMBL3225584 0.88 GRM5 (0.49) KDM4EALDH1A1HPGDHDAC1HDAC4
SCHEMBL29479790 0.86 HDAC1 (0.50) KDM4EALDH1A1HPGDHDAC1HDAC4
SCHEMBL2019162 0.84 HDAC1 (0.56) ALDH1A1HDAC1HDAC4HDAC6PARP1
SCHEMBL31298892 0.82 KDM4E (0.47) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL20028546 0.82 HDAC1 (0.58) ALDH1A1HDAC1HDAC4HDAC6PARP1
SCHEMBL16850291 0.82 HDAC1 (0.58) KDM4EHDAC1HDAC4HDAC6PARP1
SCHEMBL15120603 0.82 HDAC1 (0.55) HDAC1HDAC4HDAC6PARP1DHPS
SCHEMBL2023743 0.82 HDAC1 (0.55) HDAC1HDAC4HDAC6PARP1DHPS
SCHEMBL31666975 0.82 HDAC1 (0.60) KDM4EALDH1A1HPGDHDAC1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115843293-A Tricyclic compound, preparation method and medical application thereof 中国医药研究开发中心有限公司 2023-03-24 CN disclosed