SCHEMBL29014262

SCHEMBL29014262

COc1ccc2c(n1)NC(=O)C(NC(=O)OC(C)(C)C)CC2

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
CRBN Q96SW2 6/20 0.38
DDB1 Q16531 5/20 0.38
EPHX2 P34913 1/20 0.38
HTR2C P28335 3/20 0.37
MTNR1A P48039 3/20 0.37
MTNR1B P49286 3/20 0.37
RIPK1 Q13546 3/20 0.35
BACE1 P56817 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30314386 1.00 GAA (0.41) GAACRBNDDB1EPHX2HTR2C
SCHEMBL23900328 1.00 GAA (0.41) GAACRBNDDB1EPHX2HTR2C
SCHEMBL25875348 0.87 GAA (0.43) GAACRBNDDB1EPHX2RIPK1
SCHEMBL23887515 0.85 CRBN (0.42) CRBNDDB1HTR2CMTNR1AMTNR1B
SCHEMBL23887518 0.85 CRBN (0.42) CRBNDDB1HTR2CMTNR1AMTNR1B
SCHEMBL23555100 0.81 EPHX2 (0.46) GAACRBNDDB1EPHX2RIPK1
SCHEMBL30160156 0.81 EPHX2 (0.46) GAACRBNDDB1EPHX2RIPK1
SCHEMBL30314212 0.78 RIPK1 (0.56) RIPK1BACE1
SCHEMBL23900326 0.78 RIPK1 (0.56) RIPK1BACE1
SCHEMBL29014325 0.78 RIPK1 (0.56) RIPK1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867548-A RIP1K inhibitors 里格尔药品股份有限公司 2023-03-28 CN disclosed