SCHEMBL29017702

SCHEMBL29017702

NC(=O)Oc1ccccc1-c1ccc(N2CCCC(NC(=O)c3ccc(Br)cc3)C2)nn1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
BTK Q06187 13/20 0.40
AURKA O14965 1/20 0.40
PDPK1 O15530 1/20 0.40
AURKB Q96GD4 1/20 0.40
JAK3 P52333 6/20 0.38
MEN1 O00255 1/20 0.38
LCK P06239 3/20 0.37
EGFR P00533 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017688 0.92 BTK (0.43) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017652 0.90 BTK (0.51) BTKJAK3LCKEGFR
SCHEMBL29017672 0.90 CNR2 (0.47) KMT2ABTKJAK3MEN1LCK
SCHEMBL29637913 0.90 CNR2 (0.47) KMT2ABTKJAK3MEN1LCK
SCHEMBL29017667 0.87 AURKA (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017648 0.86 KMT2A (0.42) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017784 0.85 PPARD (0.45) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29637911 0.85 PPARD (0.45) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29637917 0.83 KMT2A (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017671 0.83 KMT2A (0.44) KMT2ABTKAURKAPDPK1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478478-B N- (1- (6- (substituted phenyl) pyridazin-3-yl) piperidin-3-yl) amine/amide derivatives and process for preparing the same 厦门大学 2023-06-13 CN disclosed