SCHEMBL29017648

SCHEMBL29017648

NC(=O)Oc1ccccc1-c1ccc(N2CCCC(NC(=O)c3ccc(Cl)c(F)c3)C2)nn1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
BTK Q06187 3/20 0.39
RORC P51449 1/20 0.39
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
DGAT2 Q96PD7 1/20 0.38
F10 P00742 1/20 0.38
AR P10275 1/20 0.37
ACHE P22303 1/20 0.37
S100A4 P26447 1/20 0.37
AURKA O14965 1/20 0.37
PDPK1 O15530 1/20 0.37
AURKB Q96GD4 1/20 0.37
JAK3 P52333 3/20 0.36
LCK P06239 2/20 0.36
EGFR P00533 1/20 0.36
USP30 Q70CQ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017688 0.89 BTK (0.43) KMT2AMEN1BTKPPARAS100A4
SCHEMBL29637977 0.89 KMT2A (0.46) KMT2AMEN1BTKRORCPPARD
SCHEMBL29017746 0.89 KMT2A (0.46) KMT2AMEN1BTKRORCPPARD
SCHEMBL29017665 0.88 KMT2A (0.44) KMT2AMEN1BTKRORCPPARD
SCHEMBL29017702 0.86 KMT2A (0.41) KMT2AMEN1BTKAURKAPDPK1
SCHEMBL29637895 0.85 PKM (0.43) KMT2AMEN1BTKPPARDPPARA
SCHEMBL29637909 0.84 MCHR1 (0.44) KMT2AMEN1BTKPPARDPPARA
SCHEMBL29017731 0.84 MCHR1 (0.44) KMT2AMEN1BTKPPARDPPARA
SCHEMBL29017652 0.84 BTK (0.51) BTKJAK3LCKEGFR
SCHEMBL29017643 0.83 MCHR1 (0.46) KMT2AMEN1BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478478-B N- (1- (6- (substituted phenyl) pyridazin-3-yl) piperidin-3-yl) amine/amide derivatives and process for preparing the same 厦门大学 2023-06-13 CN disclosed
CN-114478478-A N- (1- (6- (substituted phenyl) pyridazine-3-yl) piperidine-3-yl) amine/amide derivative and preparation method thereof 厦门大学 2022-05-13 CN disclosed