SCHEMBL29017709

SCHEMBL29017709

CNc1ccccc1-c1ccc(N2CCCC(NC(=O)c3ccc(Br)cc3)C2)nn1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
BTK Q06187 6/20 0.40
AURKA O14965 1/20 0.39
PDPK1 O15530 1/20 0.39
AURKB Q96GD4 1/20 0.39
MEN1 O00255 1/20 0.39
PPARD Q03181 2/20 0.39
PPARA Q07869 2/20 0.39
TRPV1 Q8NER1 2/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
JAK3 P52333 1/20 0.38
SYK P43405 1/20 0.37
PKM P14618 1/20 0.37
CCKAR P32238 1/20 0.36
CCKBR P32239 1/20 0.36
KCNH2 Q12809 1/20 0.36
MCHR1 Q99705 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29637984 1.00 KMT2A (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29637933 0.91 CNR1 (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017653 0.91 CNR1 (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29637945 0.90 BTK (0.51) BTKPPARDPPARAJAK3
SCHEMBL29017664 0.90 BTK (0.51) BTKPPARDPPARAJAK3
SCHEMBL29637917 0.88 KMT2A (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017671 0.88 KMT2A (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017667 0.87 AURKA (0.44) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29637911 0.87 PPARD (0.45) KMT2ABTKAURKAPDPK1AURKB
SCHEMBL29017784 0.87 PPARD (0.45) KMT2ABTKAURKAPDPK1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478478-B N- (1- (6- (substituted phenyl) pyridazin-3-yl) piperidin-3-yl) amine/amide derivatives and process for preparing the same 厦门大学 2023-06-13 CN disclosed
CN-114478478-A N- (1- (6- (substituted phenyl) pyridazine-3-yl) piperidine-3-yl) amine/amide derivative and preparation method thereof 厦门大学 2022-05-13 CN disclosed