SCHEMBL29020140

SCHEMBL29020140

CC(NC(=O)c1cc(-c2ccc(Cl)cc2)nc(-c2cnn(C)c2)n1)c1ccncc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 6/20 0.52
MAPK1 P28482 2/20 0.45
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
GSK3B P49841 2/20 0.43
WNT1 P04628 1/20 0.43
DYRK1A Q13627 1/20 0.43
THRB P10828 1/20 0.42
PDE2A O00408 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
KIT P10721 5/20 0.42
AHR P35869 1/20 0.41
ROCK2 O75116 1/20 0.40
RPS6KA5 O75582 1/20 0.40
MAP4K4 O95819 1/20 0.40
CDK1 P06493 1/20 0.40
CSF1R P07333 1/20 0.40
PRKACA P17612 1/20 0.40
FLT1 P17948 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29062372 1.00 CLK1 (0.52) CLK1MAPK1ALDH1A1MAPTGSK3B
SCHEMBL30569991 1.00 CLK1 (0.52) CLK1MAPK1ALDH1A1MAPTGSK3B
SCHEMBL29020165 0.91 CLK1 (0.52) CLK1MAPK1THRBPDE2AKIT
SCHEMBL29961629 0.91 CLK1 (0.52) CLK1MAPK1THRBPDE2AKIT
SCHEMBL29020160 0.91 CLK1 (0.52) CLK1MAPK1THRBPDE2AKIT
SCHEMBL29020182 0.90 CLK1 (0.49) CLK1MAPK1GSK3BWNT1DYRK1A
SCHEMBL29020210 0.88 CLK1 (0.48) CLK1MAPK1KITAHRROCK2
SCHEMBL29961667 0.87 CLK1 (0.50) CLK1MAPK1PDE2AKITAHR
SCHEMBL29020156 0.87 CLK1 (0.50) CLK1MAPK1PDE2AKITAHR
SCHEMBL29020159 0.87 CLK1 (0.50) CLK1MAPK1PDE2AKITAHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed