SCHEMBL29020160

SCHEMBL29020160

C[C@H](NC(=O)c1cc(-c2ccc(Cl)cc2)nc(-c2cnn(C)c2)n1)c1cnn(C)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 5/20 0.52
MAPK1 P28482 1/20 0.45
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.43
AHR P35869 1/20 0.42
THRB P10828 1/20 0.42
NAMPT P43490 1/20 0.42
PDE2A O00408 1/20 0.42
KIT P10721 4/20 0.42
EP300 Q09472 2/20 0.40
MET P08581 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020165 1.00 CLK1 (0.52) CLK1MAPK1RAB9ANPC1AHR
SCHEMBL29961629 1.00 CLK1 (0.52) CLK1MAPK1RAB9ANPC1AHR
SCHEMBL29020140 0.91 CLK1 (0.52) CLK1MAPK1AHRTHRBPDE2A
SCHEMBL29062372 0.91 CLK1 (0.52) CLK1MAPK1AHRTHRBPDE2A
SCHEMBL30569991 0.91 CLK1 (0.52) CLK1MAPK1AHRTHRBPDE2A
SCHEMBL29020156 0.90 CLK1 (0.50) CLK1MAPK1AHRPDE2AKIT
SCHEMBL29961667 0.90 CLK1 (0.50) CLK1MAPK1AHRPDE2AKIT
SCHEMBL29020159 0.90 CLK1 (0.50) CLK1MAPK1AHRPDE2AKIT
SCHEMBL29020226 0.89 MAPK1 (0.52) CLK1MAPK1PDE2AKITMET
SCHEMBL29020182 0.89 CLK1 (0.49) CLK1MAPK1AHRTHRBKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed