SCHEMBL29020155

SCHEMBL29020155

O=C(O)c1cc(-c2ccc(Cl)cc2)nc(Cl)n1.[KH]

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 4/20 0.69
MCL1 Q07820 3/20 0.60
CTRC Q99895 3/20 0.54
ALDH1A1 P00352 3/20 0.48
HPGD P15428 3/20 0.48
PTGES O14684 1/20 0.48
ALOX5 P09917 1/20 0.48
CYP2C9 P11712 1/20 0.48
CASP7 P55210 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CA12 O43570 1/20 0.47
ALPL P05186 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
DHODH Q02127 2/20 0.47
RPA1 P27694 1/20 0.44
KDM4E B2RXH2 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408569 0.98 KMO (0.71) KMOMCL1CTRCALDH1A1HPGD
Potassium SCHEMBL29961618 0.97 KMO (0.69) KMOMCL1CTRCALDH1A1HPGD
SCHEMBL29062398 0.89 KMO (0.68) KMOMCL1ALDH1A1HPGDCA12
SCHEMBL21001267 0.85 MCL1 (0.61) KMOMCL1CTRCALDH1A1HPGD
SCHEMBL34470953 0.83 MCL1 (0.60) KMOMCL1CTRCALDH1A1HPGD
SCHEMBL29020161 0.83 KMO (0.61) KMOMCL1ALDH1A1KDM4EMAPT
Potassium Ion SCHEMBL28802979 0.82 KMO (0.51) KMOMCL1CTRCALDH1A1HPGD
SCHEMBL21001316 0.81 KMO (0.67) KMOMCL1CTRCALDH1A1HPGD
SCHEMBL3408828 0.81 KMO (0.62) KMOMCL1ALDH1A1HPGDSMN1; SMN2
SCHEMBL29961681 0.80 KMO (0.56) KMOMCL1CTRCALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114835687-B AhR inhibitors 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-B AhR inhibitor, application and preparation method thereof 北京华森英诺生物科技有限公司 2023-09-05 CN disclosed
CN-115093400-A AhR inhibitor and application and preparation method thereof 重庆华森制药股份有限公司 2022-09-23 CN disclosed