SCHEMBL29020524

SCHEMBL29020524

COC(=O)c1ccc(CSc2nnc(-c3ccc(N(C)C)cc3)n2C)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.58
RAB9A P51151 3/20 0.58
HDAC3 O15379 2/20 0.58
PTK2 Q05397 2/20 0.58
HDAC1 Q13547 2/20 0.58
HDAC2 Q92769 2/20 0.58
HDAC8 Q9BY41 2/20 0.58
HDAC6 Q9UBN7 2/20 0.58
KMT2A Q03164 3/20 0.58
RGS12 O14924 1/20 0.56
ADRB2 P07550 1/20 0.56
ABL1 P00519 1/20 0.56
RIN1 Q13671 1/20 0.56
SMN1; SMN2 Q16637 6/20 0.55
TP53 P04637 1/20 0.55
MAPT P10636 4/20 0.54
MEN1 O00255 2/20 0.52
MAPK1 P28482 3/20 0.52
ALDH1A1 P00352 4/20 0.51
HPGD P15428 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4206360 0.89 HDAC2 (0.58) NPC1RAB9AHDAC2KMT2ASMN1; SMN2
SCHEMBL29020540 0.81 RGS12 (0.52) NPC1RAB9AHDAC3PTK2HDAC1
SCHEMBL29020552 0.80 NPC1 (0.56) NPC1RAB9AHDAC3PTK2HDAC1
SCHEMBL29020544 0.80 KMT2A (0.54) NPC1RAB9AHDAC3PTK2HDAC1
SCHEMBL29020522 0.77 MAPT (0.64) NPC1RAB9AKMT2ARGS12ADRB2
SCHEMBL30498865 0.77 KMT2A (0.52) NPC1RAB9AHDAC3PTK2HDAC1
SCHEMBL4216784 0.76 HDAC2 (0.61) NPC1RAB9AHDAC2KMT2ASMN1; SMN2
SCHEMBL4210891 0.75 HDAC2 (0.60) NPC1RAB9AHDAC2KMT2ASMN1; SMN2
SCHEMBL4206094 0.75 CYP3A4 (0.69) NPC1RAB9AHDAC2KMT2ASMN1; SMN2
SCHEMBL1073002 0.74 NPC1 (1.00) NPC1RAB9AKMT2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113402473-B Thiotriazole compound, preparation method and application thereof 四川省医学科学院·四川省人民医院 2023-06-23 CN disclosed
CN-113402473-A Thiotriazole compound, preparation method and application thereof 四川省医学科学院·四川省人民医院 2021-09-17 CN disclosed