SCHEMBL29020540

SCHEMBL29020540

CCC(=O)Oc1ccc(CSc2nnc(-c3ccc(N(C)C)cc3)n2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RGS12 O14924 1/20 0.52
ADRB2 P07550 1/20 0.52
NPC1 O15118 4/20 0.50
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
HDAC3 O15379 1/20 0.48
PTK2 Q05397 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PDE6D O43924 1/20 0.47
RAB9A P51151 3/20 0.47
ABL1 P00519 1/20 0.45
RIN1 Q13671 1/20 0.45
MAPT P10636 6/20 0.44
ALDH1A1 P00352 5/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HPGD P15428 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29020524 0.81 NPC1 (0.58) RGS12ADRB2NPC1KMT2AMEN1
SCHEMBL30498865 0.80 KMT2A (0.52) RGS12ADRB2NPC1KMT2AMEN1
SCHEMBL29020552 0.78 NPC1 (0.56) RGS12ADRB2NPC1KMT2AMEN1
SCHEMBL29020544 0.78 KMT2A (0.54) RGS12ADRB2NPC1KMT2AMEN1
SCHEMBL29020522 0.76 MAPT (0.64) RGS12ADRB2NPC1KMT2AMEN1
SCHEMBL4199189 0.74 CYP3A4 (0.73) NPC1KMT2AMEN1HDAC2SMN1; SMN2
SCHEMBL10621983 0.74 KMT2A (0.59) NPC1KMT2AMEN1SMN1; SMN2RAB9A
SCHEMBL4206360 0.72 HDAC2 (0.58) NPC1KMT2AMEN1HDAC2SMN1; SMN2
SCHEMBL4200573 0.70 RAB9A (0.67) NPC1KMT2AMEN1SMN1; SMN2RAB9A
SCHEMBL4206785 0.70 RAB9A (0.75) NPC1KMT2AMEN1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113402473-B Thiotriazole compound, preparation method and application thereof 四川省医学科学院·四川省人民医院 2023-06-23 CN disclosed
CN-113402473-A Thiotriazole compound, preparation method and application thereof 四川省医学科学院·四川省人民医院 2021-09-17 CN disclosed