SCHEMBL29025833

SCHEMBL29025833

CCOC(=O)C(C#N)=CNc1ccc([N+](=O)[O-])c(OCC)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.54
ALDH1A1 P00352 8/20 0.53
KDM4E B2RXH2 7/20 0.53
TDP1 Q9NUW8 1/20 0.53
MAPT P10636 3/20 0.49
LMNA P02545 3/20 0.48
NPSR1 Q6W5P4 2/20 0.48
GAA P10253 2/20 0.48
HPGD P15428 1/20 0.48
KMT2A Q03164 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
RXFP1 Q9HBX9 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
GLA P06280 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30137775 1.00 DHODH (0.54) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL22076850 0.89 DHODH (0.43) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL22076849 0.89 DHODH (0.43) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL29025829 0.89 DHODH (0.43) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL4964597 0.88 DHODH (0.57) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL18933453 0.87 DHODH (0.56) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL15223400 0.86 ALDH1A1 (0.56) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL4960852 0.83 ALDH1A1 (0.53) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL14864885 0.82 DHODH (0.46) DHODHALDH1A1KDM4ETDP1MAPT
SCHEMBL16522194 0.81 ALDH1A1 (0.59) DHODHALDH1A1KDM4ETDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109422755-B Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2023-07-04 CN disclosed
CN-109422755-A A kind of nitrogen-containing heterocycle compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2019-03-05 CN disclosed