SCHEMBL2902846

SCHEMBL2902846

CCCCC(C(O)=S)c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 4/20 0.44
KCNH2 Q12809 3/20 0.44
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 3/20 0.42
KCNE1 P15382 1/20 0.42
CYP2C19 P33261 2/20 0.42
SLC6A2 P23975 4/20 0.41
SLC6A4 P31645 4/20 0.41
CHRM2 P08172 3/20 0.41
SCN1A P35498 2/20 0.41
SCN2A Q99250 2/20 0.41
SCN3A Q9NY46 2/20 0.41
KCNJ5 P48544 1/20 0.41
KCNJ3 P48549 1/20 0.41
SCN5A Q14524 1/20 0.41
KCND3 Q9UK17 1/20 0.41
SLC6A3 Q01959 3/20 0.40
KDM4E B2RXH2 2/20 0.40
TSHR P16473 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11822611 0.86 KCNA5 (0.43) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL5669240 0.83 ALDH1A1 (0.47) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL11880698 0.81 KDM4E (0.43) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL6194668 0.80 KCNA5 (0.43) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL22610224 0.80 CYP2C19 (0.47) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL28193434 0.80 ALDH1A1 (0.49) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL1971757 0.80 TSHR (0.55) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL18601248 0.79 KCNA5 (0.42) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6
SCHEMBL9983122 0.79 ALDH1A1 (0.36) ALDH1A1CYP1A2CYP2C19SLC6A2SLC6A4
SCHEMBL11822712 0.78 KCNA5 (0.37) KCNA5KCNH2ALDH1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212305-A1 BETA-LACTONE COMPOUNDS Burnham Institute for Medical Research (US) 2010-08-04 EP disclosed
WO-2009059046-A1 BETA-LACTONE COMPOUNDS BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2009-05-07 WO disclosed