SCHEMBL29029705

SCHEMBL29029705

COC(CNc1ncnc2cc(C)c([N+](=O)[O-])cc12)OC

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.43
EGFR P00533 8/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
FBP1 P09467 1/20 0.41
PIK3CA P42336 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 2/20 0.38
HPGD P15428 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29029701 0.80 FBP1 (0.43) ABCG2EGFRFBP1ALDH1A1HTT
SCHEMBL8932207 0.79 EGFR (0.50) ABCG2EGFRFBP1
SCHEMBL29361152 0.73 PIK3CA (0.61) MEN1KMT2APIK3CAALDH1A1HTT
SCHEMBL20412178 0.72 GAA (0.44) ABCG2EGFRMEN1KMT2AFBP1
SCHEMBL14579636 0.71 GAA (0.43) ABCG2EGFRMEN1KMT2AALDH1A1
SCHEMBL7474113 0.70 EGFR (0.55) ABCG2EGFRFBP1ALDH1A1KDM4E
SCHEMBL8825777 0.70 EGFR (0.50) ABCG2EGFRFBP1
SCHEMBL14579634 0.70 GAA (0.42) ABCG2EGFRMEN1KMT2AALDH1A1
SCHEMBL28755534 0.70 GAA (0.49) EGFRKMT2AALDH1A1HTT
SCHEMBL28821207 0.70 CCNC (0.38) EGFRMEN1KMT2AFBP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116406272-A DNA-PK selective inhibitor and preparation method and application thereof 首药控股(北京)股份有限公司 2023-07-07 CN disclosed
CN-114605414-A DNA-PK selective inhibitor and preparation method and application thereof 首药控股(北京)股份有限公司 2022-06-10 CN disclosed
WO-2022017368-A1 DNA-PK SELECTIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 首药控股(北京)股份有限公司 2022-01-27 WO disclosed