SCHEMBL29030477

SCHEMBL29030477

C#Cc1ccc(-c2nnc(NC3CCCN(C(=O)OC(C)(C)C)C3)nc2OC)c(OCOCC)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 2/20 0.40
EHMT2 Q96KQ7 1/20 0.37
MERTK Q12866 1/20 0.37
PIK3CD O00329 2/20 0.36
USP30 Q70CQ3 2/20 0.36
TRPV1 Q8NER1 1/20 0.36
SUV39H2 Q9H5I1 1/20 0.35
PIM1 P11309 2/20 0.35
PIM2 Q9P1W9 2/20 0.35
HDAC4 P56524 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
BRD4 O60885 1/20 0.34
CCNK O75909 1/20 0.34
CDK12 Q9NYV4 1/20 0.34
PIK3CA P42336 1/20 0.34
NSD2 O96028 1/20 0.34
PARP1 P09874 1/20 0.34
DNMT3A Q9Y6K1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30488497 1.00 BTK (0.40) BTKEHMT2MERTKPIK3CDUSP30
SCHEMBL25295324 1.00 BTK (0.40) BTKEHMT2MERTKPIK3CDUSP30
SCHEMBL30833925 0.92 BTK (0.41) BTKEHMT2MERTKUSP30TRPV1
SCHEMBL30893689 0.92 BTK (0.41) BTKEHMT2MERTKUSP30TRPV1
SCHEMBL30833985 0.91 BTK (0.40) BTKEHMT2MERTKUSP30TRPV1
SCHEMBL30517816 0.91 CCNK (0.36) CCNKCDK12
SCHEMBL29030536 0.90 BTK (0.40) BTKEHMT2MERTKUSP30TRPV1
SCHEMBL30488580 0.90 BTK (0.40) BTKEHMT2MERTKUSP30TRPV1
SCHEMBL29030534 0.90 BTK (0.40) BTKEHMT2MERTKUSP30TRPV1
SCHEMBL30893688 0.86 NLRP3 (0.46) EHMT2USP30PIM1PIM2BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116410140-A NLRP3 inflammation corpuscle inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2023-07-11 CN disclosed