SCHEMBL29031963

SCHEMBL29031963

Cc1cc(Cn2ncc3c(-c4ccncc4)nc(N)nc32)ccc1N

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.49
ADORA1 P30542 15/20 0.49
ADORA3 P0DMS8 1/20 0.46
ADORA2B P29275 1/20 0.46
HDAC1 Q13547 3/20 0.43
HSP90AA1 P07900 1/20 0.43
TRAP1 Q12931 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
ATM Q13315 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29616973 0.85 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL23388322 0.85 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29031953 0.84 ADORA2A (0.52) ADORA2AADORA1HDAC1HSP90AA1TRAP1
SCHEMBL29617002 0.83 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL23388284 0.83 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29616994 0.83 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29031965 0.82 ADORA2A (0.62) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL23388312 0.81 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29617020 0.81 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29617022 0.81 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116425756-A Adenosine receptor antagonist compounds and uses thereof 日东制药株式会社 2023-07-14 CN disclosed