SCHEMBL29037148

SCHEMBL29037148

COc1ccc(Cn2cnc3c(Nc4ccnc5ccccc45)nc(-c4cccc(C)n4)nc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 11/20 0.50
TGFBR2 P37173 1/20 0.50
HTT P42858 1/20 0.43
CTSL P07711 2/20 0.43
HDAC1 Q13547 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
PDGFRA P16234 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
YTHDC1 Q96MU7 1/20 0.40
ADORA2A P29274 2/20 0.40
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18554152 0.84 TGFBR1 (0.50) TGFBR1TGFBR2CTSLHDAC1HDAC3
SCHEMBL18554366 0.81 CCNE1 (0.48) TGFBR1CTSLHDAC1HDAC3HDAC2
SCHEMBL18554274 0.78 TGFBR1 (0.53) TGFBR1TGFBR2HDAC1HDAC3HDAC2
SCHEMBL22978902 0.78 ADORA2A (0.46) CTSLHDAC1HDAC2PDGFRACCNE1
SCHEMBL29365625 0.78 ADORA2A (0.46) CTSLHDAC1HDAC2PDGFRACCNE1
SCHEMBL29366198 0.76 HPGD (0.58) HTTCTSLHDAC1HDAC3HDAC2
SCHEMBL18554153 0.76 HPGD (0.58) HTTCTSLHDAC1HDAC3HDAC2
SCHEMBL18554142 0.76 TGFBR1 (0.44) TGFBR1CTSLHDAC1HDAC3HDAC2
SCHEMBL18554195 0.76 TGFBR1 (0.52) TGFBR1TGFBR2CTSLHDAC1HDAC3
SCHEMBL18554354 0.75 BUB1 (0.51) TGFBR1TGFBR2CTSLHDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116789681-A Imidazo pyrimidine compound containing fused ring group, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-09-22 CN disclosed
CN-112341477-B Imidazo pyrimidine compound containing fused ring group, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-07-21 CN disclosed
CN-112341477-A Imidazo pyrimidine compound containing polycyclic group, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-02-09 CN disclosed