SCHEMBL29037239

SCHEMBL29037239

CC(C)COc1ccc(CN(Cc2ccn(C)n2)C(=O)CC2CCN(C)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 20/20 0.55
HTR2C P28335 4/20 0.55
ABCB11 O95342 1/20 0.47
CYP1A2 P05177 1/20 0.47
ADRB2 P07550 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD1 P21728 1/20 0.47
TBXA2R P21731 1/20 0.47
SLC6A2 P23975 1/20 0.47
GPR183 P32249 1/20 0.47
CYP2C19 P33261 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
APLNR P35414 1/20 0.47
DRD3 P35462 1/20 0.47
CX3CR1 P49238 1/20 0.47
SLC6A3 Q01959 1/20 0.47
KCNH2 Q12809 1/20 0.47
GPR65 Q8IYL9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25466903 0.78 HTR2A (0.79) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20767191 0.76 HTR2A (0.57) HTR2ACHRM1OPRM1HRH3
SCHEMBL20766900 0.76 HTR2A (0.68) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20766920 0.75 HTR2A (0.56) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20781016 0.74 HTR2A (0.65) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20781090 0.73 HTR2A (0.56) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL30504379 0.73 HTR2A (0.54) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20766953 0.72 HTR2A (0.68) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20767249 0.72 HTR2A (0.52) HTR2AHTR2CABCB11CYP1A2ADRB2
SCHEMBL20766869 0.72 HTR2A (0.50) HTR2AHTR2CABCB11CYP1A2ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549006-A Amide derivative and application thereof 江苏恩华药业股份有限公司 2021-10-26 CN claimed
CN-113549006-B Amide derivative and application thereof 江苏恩华药业股份有限公司 2023-07-21 CN disclosed
CN-113549006-A Amide derivative and application thereof 江苏恩华药业股份有限公司 2021-10-26 CN disclosed