SCHEMBL29037792

SCHEMBL29037792

COc1cccc(F)c1C(=O)Nc1nc(Cl)ncc1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.50
SRC P12931 1/20 0.50
POLB P06746 1/20 0.46
BCR P11274 1/20 0.45
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
KMT2A Q03164 4/20 0.42
RAB9A P51151 2/20 0.42
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41
MEN1 O00255 3/20 0.41
HCRTR1 O43613 2/20 0.41
GAA P10253 2/20 0.41
HCRTR2 O43614 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
RECQL P46063 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29520601 0.89 ABL1 (0.52) ABL1SRCPOLBCCNA2CDK2
SCHEMBL29037823 0.89 ABL1 (0.52) ABL1SRCPOLBCCNA2CDK2
SCHEMBL29037737 0.84 SRC (0.48) ABL1SRCPOLBCCNA2CDK2
SCHEMBL29520459 0.84 SRC (0.48) ABL1SRCPOLBCCNA2CDK2
SCHEMBL29037797 0.78 ABL1 (0.45) ABL1SRCPOLBKMT2ARAB9A
SCHEMBL29520398 0.78 ABL1 (0.45) ABL1SRCPOLBKMT2ARAB9A
SCHEMBL29037765 0.72 IL2 (0.39) ABL1SRCPOLBBCRCCNA2
SCHEMBL29520303 0.72 IL2 (0.39) ABL1SRCPOLBBCRCCNA2
SCHEMBL6989383 0.72 KMT2A (0.59) ABL1SRCPOLBKMT2ARAB9A
SCHEMBL22500906 0.71 ABL1 (0.47) ABL1BCRCDK2KMT2AAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116456985-A Pyrimidine and pyridine derivatives as HPK1 modulators and methods of use thereof 深圳市原力生命科学有限公司 2023-07-18 CN disclosed
WO-2022063140-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AS HPK1 MODULATOR AND METHODS USING SAME SHENZHEN IONOVA LIFE SCIENCE CO., LTD. (CN) 2022-03-31 WO disclosed