SCHEMBL29520303

SCHEMBL29520303

C=CCOc1cccc(F)c1C(=O)Nc1nc(Cl)ncc1C=C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL2 P60568 1/20 0.39
ALDH1A1 P00352 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LIG1 P18858 1/20 0.38
ABL1 P00519 2/20 0.37
SRC P12931 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNQ3 O43525 2/20 0.36
KCNQ2 O43526 2/20 0.36
KCNQ5 Q9NR82 2/20 0.36
MAOB P27338 1/20 0.35
NPC1 O15118 1/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29037765 1.00 IL2 (0.39) IL2ALDH1A1L3MBTL1LIG1ABL1
SCHEMBL29037800 0.78 IL2 (0.40) IL2L3MBTL1LIG1ABL1SRC
SCHEMBL29037823 0.74 ABL1 (0.52) ALDH1A1ABL1SRCMEN1KMT2A
SCHEMBL29520601 0.74 ABL1 (0.52) ALDH1A1ABL1SRCMEN1KMT2A
SCHEMBL29037792 0.72 ABL1 (0.50) ALDH1A1ABL1SRCMEN1KMT2A
SCHEMBL2061375 0.72 L3MBTL1 (0.43) ALDH1A1L3MBTL1
SCHEMBL29037809 0.71 LIG1 (0.47) IL2ALDH1A1L3MBTL1LIG1MEN1
SCHEMBL29520459 0.70 SRC (0.48) ABL1SRCMEN1KMT2ANPC1
SCHEMBL29037737 0.70 SRC (0.48) ABL1SRCMEN1KMT2ANPC1
SCHEMBL15867225 0.69 CYP3A4 (0.49) IL2ALDH1A1L3MBTL1LIG1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116456985-A Pyrimidine and pyridine derivatives as HPK1 modulators and methods of use thereof 深圳市原力生命科学有限公司 2023-07-18 CN disclosed
WO-2022063140-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AS HPK1 MODULATOR AND METHODS USING SAME SHENZHEN IONOVA LIFE SCIENCE CO., LTD. (CN) 2022-03-31 WO disclosed