SCHEMBL29042018

SCHEMBL29042018

Brc1ccc2c(cnn2C2CCN(C3CCOCC3)CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 5/20 0.42
IRAK4 Q9NWZ3 2/20 0.40
PDE4D Q08499 2/20 0.40
MAPK1 P28482 2/20 0.39
CHRM2 P08172 2/20 0.37
CHRM4 P08173 2/20 0.37
CHRM1 P11229 2/20 0.37
CHRM5 P08912 1/20 0.37
CHRM3 P20309 1/20 0.37
KCNH2 Q12809 1/20 0.37
LRRK2 Q5S007 1/20 0.37
PDE1A P54750 2/20 0.36
PDE1B Q01064 2/20 0.36
PDE1C Q14123 2/20 0.36
WNT1 P04628 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
SCD O00767 1/20 0.36
MBTD1 Q05BQ5 1/20 0.36
L3MBTL3 Q96JM7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29041986 0.93 PIK3CD (0.41) PIK3CDIRAK4PDE4DMAPK1CHRM2
SCHEMBL29042117 0.93 PIK3CD (0.41) PIK3CDIRAK4PDE4DMAPK1CHRM2
SCHEMBL30122245 0.92 PIK3CD (0.47) PIK3CDPDE4DMAPK1PDE1APDE1B
SCHEMBL29041973 0.89 LRRK2 (0.40) PIK3CDKCNH2LRRK2WNT1GSK3B
SCHEMBL26757187 0.84 PIK3CD (0.40) PIK3CDPDE4DMAPK1PDE1APDE1B
SCHEMBL21175144 0.84 PIK3CD (0.40) PIK3CDPDE4DMAPK1PDE1APDE1B
SCHEMBL20014996 0.84 PIK3CD (0.40) PIK3CDPDE4DMAPK1PDE1APDE1B
SCHEMBL29042016 0.83 SCD (0.37) CHRM1KCNH2SCDMBTD1L3MBTL3
SCHEMBL13468 0.82 HDAC8 (0.39) PIK3CDKCNH2SCD
SCHEMBL19279630 0.81 PIK3CD (0.55) PIK3CDPDE4DMAPK1PDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed