SCHEMBL29042016

SCHEMBL29042016

FC1(F)CCC(N2CCC(n3ncc4cc(Br)ccc43)CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.37
HTR2A P28223 5/20 0.37
HTR7 P34969 5/20 0.37
KCNH2 Q12809 3/20 0.37
DRD2 P14416 3/20 0.35
MBTD1 Q05BQ5 1/20 0.34
L3MBTL3 Q96JM7 1/20 0.34
PARP1 P09874 7/20 0.34
PARP2 Q9UGN5 4/20 0.34
GPR119 Q8TDV5 2/20 0.34
CHRM1 P11229 1/20 0.34
KDM5A P29375 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
TEAD1 P28347 1/20 0.33
TEAD4 Q15561 1/20 0.33
TEAD2 Q15562 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2B6 P20813 1/20 0.32
HTR1A P08908 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29042018 0.83 PIK3CD (0.42) SCDKCNH2MBTD1L3MBTL3CHRM1
SCHEMBL31482815 0.82 KMO (0.40) SCDKDM5AKDM4CKDM5BTEAD1
SCHEMBL29041973 0.81 LRRK2 (0.40) SCDKCNH2GPR119
SCHEMBL13468 0.80 HDAC8 (0.39) SCDHTR2AHTR7KCNH2DRD2
SCHEMBL30613532 0.79 IRAK4 (0.37) SCDHTR2AHTR7KCNH2DRD2
SCHEMBL29041994 0.79 IRAK4 (0.37) SCDHTR2AHTR7KCNH2DRD2
SCHEMBL26683794 0.78 HTR1A (0.46) SCDHTR2AHTR7KCNH2DRD2
SCHEMBL25045382 0.78 HTR7 (0.39) SCDHTR2AHTR7KCNH2GPR119
SCHEMBL17678127 0.78 PDE9A (0.38) SCDHTR2AHTR7KCNH2DRD2
SCHEMBL29042132 0.78 HTR7 (0.41) SCDHTR2AHTR7KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
WO-2023198114-A1 ALK2 KINASE INHIBITOR 杭州邦顺制药有限公司 2023-10-19 WO disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed