SCHEMBL2904415

SCHEMBL2904415

Nc1nc(NCCCn2cc(C(=O)N3CCC(NC(=O)C(F)(F)F)C3)c(-c3ccc(-n4ccnc4)cc3)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
CD38 P28907 8/20 0.33
PIK3CD O00329 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2911578 0.92 GSK3A (0.38) CDK1GSK3AGSK3BCD38PIK3CD
SCHEMBL2904171 0.92 GSK3A (0.38) CDK1GSK3AGSK3BCD38PIK3CD
SCHEMBL2906860 0.87 GSK3A (0.39) CDK1GSK3AGSK3BPIK3CD
SCHEMBL2909976 0.86 GSK3A (0.39) CDK1GSK3AGSK3B
SCHEMBL2913331 0.85 CDK1 (0.41) CDK1GSK3AGSK3BCD38
SCHEMBL2909662 0.82 GSK3A (0.44) CDK1GSK3AGSK3B
SCHEMBL2909762 0.81 CDK1 (0.38) CDK1GSK3AGSK3BCD38
SCHEMBL2910066 0.81 GSK3A (0.38) CDK1GSK3AGSK3BCD38
SCHEMBL2903761 0.81 CDK1 (0.38) CDK1GSK3AGSK3BCD38
SCHEMBL2912012 0.80 GSK3A (0.41) CDK1GSK3AGSK3BPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed