SCHEMBL2904464

SCHEMBL2904464

O=C(/C=C/c1ccc(F)c(Cl)c1)N1CCC(=O)N(CCCCN2CCN(C3CCCC3)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PYGL P06737 7/20 0.46
GPR183 P32249 2/20 0.44
CCR2 P41597 2/20 0.43
ITGB2 P05107 1/20 0.40
ICAM1 P05362 1/20 0.40
ITGAL P20701 1/20 0.40
SLC2A1 P11166 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904466 1.00 PYGL (0.46) PYGLGPR183CCR2ITGB2ICAM1
SCHEMBL2904453 0.97 PYGL (0.47) PYGLGPR183CCR2SLC2A1
SCHEMBL2904455 0.97 PYGL (0.47) PYGLGPR183CCR2SLC2A1
SCHEMBL2903668 0.93 GPR183 (0.50) PYGLGPR183CCR2SLC2A1
SCHEMBL2903314 0.93 GPR183 (0.50) PYGLGPR183CCR2SLC2A1
SCHEMBL2904897 0.91 GPR183 (0.50) PYGLGPR183CCR2SLC2A1
SCHEMBL2904898 0.91 GPR183 (0.50) PYGLGPR183CCR2SLC2A1
SCHEMBL2899068 0.89 GPR183 (0.52) PYGLGPR183CCR2SLC2A1
SCHEMBL2899072 0.89 GPR183 (0.52) PYGLGPR183CCR2SLC2A1
SCHEMBL2897821 0.89 PYGL (0.50) PYGLGPR183CCR2ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed