SCHEMBL2904491

SCHEMBL2904491

O=C(/C=C/c1ccc(F)c(Cl)c1)N1CCC(=O)N(CCCN2CC[C@@H](CO)[C@@H](O)C2)CC1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 6/20 0.41
GPR183 P32249 3/20 0.40
PYGL P06737 2/20 0.40
ITGB2 P05107 2/20 0.37
ICAM1 P05362 2/20 0.37
ITGAL P20701 2/20 0.37
SLC2A1 P11166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2899434 0.93 CCR2 (0.47) CCR2GPR183PYGLSLC2A1
SCHEMBL2899436 0.93 CCR2 (0.47) CCR2GPR183PYGLSLC2A1
SCHEMBL2903082 0.93 CCR2 (0.47) CCR2GPR183PYGLSLC2A1
SCHEMBL2902267 0.92 CCR2 (0.40) CCR2GPR183PYGLITGB2ICAM1
SCHEMBL2899274 0.91 CCR2 (0.47) CCR2GPR183PYGLSLC2A1
SCHEMBL2902728 0.91 CCR2 (0.47) CCR2GPR183PYGLSLC2A1
SCHEMBL2903003 0.91 CCR2 (0.42) CCR2GPR183PYGLITGB2ICAM1
SCHEMBL2903001 0.91 CCR2 (0.42) CCR2GPR183PYGLITGB2ICAM1
SCHEMBL2899701 0.90 CCR2 (0.42) CCR2GPR183PYGLITGB2ICAM1
SCHEMBL2897579 0.89 CCR2 (0.42) CCR2GPR183PYGLITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed