SCHEMBL2904548

SCHEMBL2904548

COC[C@H]1CCN(C[C@H](O)CN2CCN(C(=O)C=Cc3ccc(Cl)c(Cl)c3)CCC2=O)C[C@H]1O

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 10/20 0.44
GPR183 P32249 5/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SLC2A1 P11166 1/20 0.39
KDM4E B2RXH2 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904543 1.00 CCR2 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2904546 1.00 CCR2 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2902597 0.95 CCR2 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2899761 0.93 CCR2 (0.38) CCR2GPR183KDM4ECYP3A4HPGD
SCHEMBL2899760 0.93 CCR2 (0.38) CCR2GPR183KDM4ECYP3A4HPGD
SCHEMBL2899757 0.93 CCR2 (0.38) CCR2GPR183KDM4ECYP3A4HPGD
SCHEMBL2898703 0.92 CCR2 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2904095 0.92 GPR183 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2904092 0.92 GPR183 (0.44) CCR2GPR183NPC1RAB9ATDP1
SCHEMBL2902522 0.92 GPR183 (0.44) CCR2GPR183NPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed