SCHEMBL29045900

SCHEMBL29045900

CC(=O)N[C@H](C)c1nccc2c1[nH]c1ccc(Br)cc12

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
DYRK1A Q13627 1/20 0.40
ACACB O00763 1/20 0.40
CHUK O15111 1/20 0.40
BRAF P15056 2/20 0.39
KIT P10721 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
PARP14 Q460N5 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PIM3 Q86V86 2/20 0.38
BAZ2B Q9UIF8 2/20 0.38
ERBB2 P04626 1/20 0.38
PIM1 P11309 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29986202 1.00 AR (0.42) ARRXFP1DYRK1AACACBCHUK
SCHEMBL29045902 1.00 AR (0.42) ARRXFP1DYRK1AACACBCHUK
SCHEMBL29045928 0.92 DYRK1A (0.47) DYRK1AACACBPARP14PIM3L3MBTL1
SCHEMBL29045926 0.92 DYRK1A (0.47) DYRK1AACACBPARP14PIM3L3MBTL1
SCHEMBL29986906 0.87 BCHE (0.49) RXFP1DYRK1ABRAFPARP14L3MBTL1
SCHEMBL29045894 0.87 HTR2C (0.44) DYRK1ABRAFKITPARP14ERBB2
SCHEMBL29045890 0.87 HTR2C (0.44) DYRK1ABRAFKITPARP14ERBB2
SCHEMBL29045901 0.87 BCHE (0.49) RXFP1DYRK1ABRAFPARP14L3MBTL1
SCHEMBL29986612 0.87 HTR2C (0.44) DYRK1ABRAFKITPARP14ERBB2
SCHEMBL29045899 0.87 BCHE (0.49) RXFP1DYRK1ABRAFPARP14L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304597-B Beta-carboline compounds and application thereof in preparation of medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2023-10-20 CN disclosed
CN-115304597-A Beta-carboline compounds and application thereof in preparing medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2022-11-08 CN disclosed