SCHEMBL29045926

SCHEMBL29045926

CC(=O)N[C@H](C)c1nccc2c1[nH]c1cc(Br)ccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 7/20 0.47
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
ROCK2 O75116 2/20 0.41
ACACB O00763 1/20 0.39
PARP14 Q460N5 1/20 0.38
MAOA P21397 2/20 0.38
PIM3 Q86V86 1/20 0.38
CYP1A2 P05177 1/20 0.38
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
CCNA1 P78396 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
GSK3B P49841 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29045928 1.00 DYRK1A (0.47) DYRK1ABCHEACHEROCK2ACACB
SCHEMBL29045902 0.92 AR (0.42) DYRK1AACACBPARP14PIM3L3MBTL1
SCHEMBL29986202 0.92 AR (0.42) DYRK1AACACBPARP14PIM3L3MBTL1
SCHEMBL29045900 0.92 AR (0.42) DYRK1AACACBPARP14PIM3L3MBTL1
SCHEMBL29045942 0.86 DYRK1A (0.43) DYRK1ABCHEACHEROCK2PARP14
SCHEMBL29045951 0.83 PARP14 (0.54) DYRK1ABCHEPARP14MAOACYP1A2
SCHEMBL29045946 0.83 PARP14 (0.54) DYRK1ABCHEPARP14MAOACYP1A2
SCHEMBL29045899 0.81 BCHE (0.49) DYRK1ABCHEACHEROCK2PARP14
SCHEMBL29986906 0.81 BCHE (0.49) DYRK1ABCHEACHEROCK2PARP14
SCHEMBL29045894 0.81 HTR2C (0.44) DYRK1ABCHEACHEROCK2PARP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304597-B Beta-carboline compounds and application thereof in preparation of medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2023-10-20 CN disclosed
CN-115304597-A Beta-carboline compounds and application thereof in preparing medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2022-11-08 CN disclosed