SCHEMBL29045951

SCHEMBL29045951

CC(=O)NC(C)c1nccc2c1[nH]c1ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP14 Q460N5 2/20 0.54
KDM4E B2RXH2 4/20 0.50
TDO2 P48775 3/20 0.50
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
MAPT P10636 2/20 0.50
MAPK1 P28482 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
GABRP O00591 1/20 0.50
GABRD O14764 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
GABRA1 P14867 1/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
GABRB1 P18505 1/20 0.50
GABRG2 P18507 1/20 0.50
NFKB1 P19838 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29045946 1.00 PARP14 (0.54) PARP14KDM4ETDO2KMT2AMEN1
SCHEMBL29045922 0.89 PARP14 (0.53) PARP14KDM4ETDO2KMT2AMEN1
SCHEMBL29045932 0.87 BCHE (0.46) PARP14TDO2KMT2AMEN1GABRA1
SCHEMBL29986196 0.87 BCHE (0.46) PARP14TDO2KMT2AMEN1GABRA1
SCHEMBL29045936 0.87 BCHE (0.46) PARP14TDO2KMT2AMEN1GABRA1
SCHEMBL29045899 0.85 BCHE (0.49) PARP14KDM4EMAPTALDH1A1BCHE
SCHEMBL29986906 0.85 BCHE (0.49) PARP14KDM4EMAPTALDH1A1BCHE
SCHEMBL29045894 0.85 HTR2C (0.44) PARP14GABRPGABRDGABRA1GABRB1
SCHEMBL29045901 0.85 BCHE (0.49) PARP14KDM4EMAPTALDH1A1BCHE
SCHEMBL29986612 0.85 HTR2C (0.44) PARP14GABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304597-B Beta-carboline compounds and application thereof in preparation of medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2023-10-20 CN disclosed
CN-115304597-A Beta-carboline compounds and application thereof in preparing medicines for treating or preventing tumor diseases 中国科学院深圳先进技术研究院 2022-11-08 CN disclosed